Toradol Medication for Pain Relief
Updated in July 2021
Toradol is a non-steroidal anti-inflammatory drug that is used to treat moderate to severe pain, inflammation, and fever. The active ingredient in Toradol is ketorolac tromethamine. It is a racemic blend of [-] S- and also [+] R-enantiomeric kinds, with the S-form having analgesic activity.
At higher doses, there is a proportional increase in the concentration of free and bound racemate. It works by blocking the production of certain natural substances in the body that cause pain and inflammation. The drug is available in the form of a tablet, injection, or nasal spray, and is usually given in a hospital setting or doctor's office.
About 92% of a given dosage is found in the urine, around 40% as metabolites and 60% as unmodified ketorolac.